| # | Country | Total Patents | |
|---|---|---|---|
| #1 | EPO (European Patent Office) | 13 | |
| #2 | Australia | 10 | |
| #3 | United States | 10 | |
| #4 | Israel | 6 | |
| #5 | Singapore | 4 | |
| #6 | Brazil | 3 | |
| #7 | Canada | 3 | |
| #8 | Republic of Korea | 3 | |
| #9 | WIPO (World Intellectual Property Organization) | 3 | |
| #10 | Chile | 2 | |
| #11 | Hong Kong | 2 | |
| #12 | Mexico | 2 | |
| #13 | Russian Federation | 2 | |
| #14 | Taiwan | 2 | |
| #15 | Colombia | 1 | |
| #16 | Ecuador | 1 | |
| #17 | Hungary | 1 | |
| #18 | Jordan | 1 | |
| #19 | Japan | 1 | |
| #20 | Morocco | 1 | |
| #21 | Peru | 1 | |
| #22 | Philippines | 1 | |
| #23 | Serbia | 1 | |
| #24 | Ukraine | 1 |
| # | Industry | |
|---|---|---|
| #1 | Pharmaceuticals | |
| #2 | Organic fine chemistry | |
| #3 | Biotechnology |
| # | Technology | |
|---|---|---|
| #1 | Heterocyclic compounds | |
| #2 | Therapeutic chemical compounds | |
| #3 | Medical preparations | |
| #4 | Organic chemistry methods | |
| #5 | Peptides | |
| #6 | Acyclic or carbocyclic compounds |
| # | Name | Total Patents |
|---|---|---|
| #1 | Zhai Dayong | 59 |
| #2 | Rogers Evan W | 57 |
| #3 | Cui Jingrong Jean | 50 |
| #4 | Deng Wei | 35 |
| #5 | Ung Jane | 32 |
| #6 | Li Yishan | 28 |
| #7 | Zhang Han | 24 |
| #8 | Whitten Jeffrey | 23 |
| #9 | Huang Zhongdong | 16 |
| #10 | Cui Jingrong J | 11 |
| Publication | Filing date | Title |
|---|---|---|
| WO2020257165A1 | Macrocycles for use in treating disease | |
| WO2020257189A1 | Macrocycles for treating disease | |
| WO2020257169A1 | Polymorphs of a macrocyclic kinase inhibitor | |
| EP3728271A1 | Macrocyclic compounds for treating disease | |
| MA49994A1 | Macrocyclic compounds for the treatment of disease | |
| TW201612183A | Diaryl macrocycles as modulators of protein kinases |