| # | Country | Total Patents | |
|---|---|---|---|
| #1 | China | 10 | |
| #2 | WIPO (World Intellectual Property Organization) | 9 | |
| #3 | United States | 7 | |
| #4 | Taiwan | 6 | |
| #5 | Canada | 5 | |
| #6 | Republic of Korea | 5 | |
| #7 | Mexico | 4 | |
| #8 | Brazil | 3 | |
| #9 | Israel | 3 | |
| #10 | African Regional Industrial Property Organization | 2 | |
| #11 | Singapore | 2 | |
| #12 | South Africa | 2 | |
| #13 | Argentina | 1 | |
| #14 | Chile | 1 | |
| #15 | EAPO (Eurasian Patent Organization) | 1 | |
| #16 | EPO (European Patent Office) | 1 | |
| #17 | Hong Kong | 1 | |
| #18 | Peru | 1 | |
| #19 | Philippines | 1 |
| # | Industry | |
|---|---|---|
| #1 | Pharmaceuticals | |
| #2 | Organic fine chemistry | |
| #3 | Biotechnology |
| # | Technology | |
|---|---|---|
| #1 | Therapeutic chemical compounds | |
| #2 | Heterocyclic compounds | |
| #3 | Medical preparations | |
| #4 | Organic chemistry methods | |
| #5 | Acyclic or carbocyclic compounds | |
| #6 | Peptides |
| # | Name | Total Patents |
|---|---|---|
| #1 | Rogers Evan W | 48 |
| #2 | Zhai Dayong | 46 |
| #3 | Cui Jingrong Jean | 37 |
| #4 | Li Yishan | 35 |
| #5 | Ung Jane | 21 |
| #6 | Deng Wei | 20 |
| #7 | Cui Jingrong J | 14 |
| #8 | Evan W Rogers | 10 |
| #9 | Zhang Han | 8 |
| #10 | Whitten Jeffrey | 8 |
| Publication | Filing date | Title |
|---|---|---|
| WO2019126122A1 | Macrocyclic kinase inhibitors and their use | |
| CN111182903A | Macrocyclic compounds and uses thereof | |
| TW201831188A | Combination therapy involving diaryl macrocyclic compounds | |
| CN109715165A | Huge ring kinase inhibitor | |
| KR20180033194A | Chiral Diaryl Macrocycles and Their Uses | |
| CN108026108A | diaryl macrocyclic polymorphs | |
| US2018186813A1 | Chiral diaryl macrocycles as modulators of protein kinases | |
| CN106170289A | The huge ring of diaryl as the regulator of protein kinase |